Solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones

Blanca Martínez-Teipel; Enrique Michelotti; Martha J. Kelly; Damian G. Weaver; Francis Acholla; Kebede Beshah; Jordi Teixidó

doi:10.1016/S0040-4039(01)01095-4

Solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones

Blanca Martínez-Teipel^*
, Enrique Michelotti
, Martha J. Kelly
, Damian G. Weaver
, Francis Acholla
, Kebede Beshah
, Jordi Teixidó

^*Corresponding author for this work

Research output: Indexed journal article › Article › peer-review

12 Citations (Scopus)

Abstract

The solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones from imidate esters and substituted hydrazines is reported. The synthesis starts with the reaction of imidic esters with polymer-bound glycine to form the imidate esters. A rehearsal library of 59 compounds was synthesized.

Original language	English
Pages (from-to)	6455-6457
Number of pages	3
Journal	Tetrahedron Letters
Volume	42
Issue number	37
DOIs	https://doi.org/10.1016/S0040-4039(01)01095-4
Publication status	Published - 10 Sept 2001

Keywords

Dihydro-1,2,4-triazin-6(1h)-ones

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10.1016/S0040-4039(01)01095-4

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title = "Solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones",

abstract = "The solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones from imidate esters and substituted hydrazines is reported. The synthesis starts with the reaction of imidic esters with polymer-bound glycine to form the imidate esters. A rehearsal library of 59 compounds was synthesized.",

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doi = "10.1016/S0040-4039(01)01095-4",

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T1 - Solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones

AU - Martínez-Teipel, Blanca

AU - Michelotti, Enrique

AU - Kelly, Martha J.

AU - Weaver, Damian G.

AU - Acholla, Francis

AU - Beshah, Kebede

AU - Teixidó, Jordi

PY - 2001/9/10

Y1 - 2001/9/10

N2 - The solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones from imidate esters and substituted hydrazines is reported. The synthesis starts with the reaction of imidic esters with polymer-bound glycine to form the imidate esters. A rehearsal library of 59 compounds was synthesized.

AB - The solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones from imidate esters and substituted hydrazines is reported. The synthesis starts with the reaction of imidic esters with polymer-bound glycine to form the imidate esters. A rehearsal library of 59 compounds was synthesized.

KW - Dihydro-1,2,4-triazin-6(1h)-ones

UR - https://www.scopus.com/pages/publications/0035840371

UR - https://www.webofscience.com/api/gateway?GWVersion=2&SrcApp=pure_univeritat_ramon_llull&SrcAuth=WosAPI&KeyUT=WOS:000170753900007&DestLinkType=FullRecord&DestApp=WOS_CPL

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M3 - Article

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SN - 0040-4039

VL - 42

SP - 6455

EP - 6457

JO - Tetrahedron Letters

JF - Tetrahedron Letters

IS - 37

ER -

Solid-phase synthesis of 1-substituted 4,5-dihydro-1,2,4-triazin-6-ones

Abstract

Keywords

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