Structure-Based Discovery of Proline-Derived Arginase Inhibitors with Improved Oral Bioavailability for Immuno-Oncology

Min Lu, Hongjun Zhang, Derun Li, Matthew Childers, Qinglin Pu, Rachel L. Palte, Symon Gathiaka, Thomas W. Lyons, Anandan Palani, Peter W. Fan, Peter Spacciapoli, J. Richard Miller, Hyelim Cho, Mangeng Cheng, Kalyan Chakravarthy, Jennifer O'Neil, Padmanabhan Eangoor, Adam Beard, Hai-Young Kim, Josep SauriHakan Gunaydin, David L. Sloman, Phieng Siliphaivanh, Jared Cumming, Christian Fischer

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Pharmacology, Toxicology and Pharmaceutical Science