Cyclization of tautomeric 1,5-dinitrile systems with hydrogen halides: A definitive mechanistic rationalization?

Jordi Teixidó, José I. Borrell, Blanca Serra, Josep Lluis Matallana, Carles Colominas, Francisco Carrión, Rosalia Pascual, Josep Lluis Falcó, Xavier Batllori

Producció científica: Article en revista indexadaArticleAvaluat per experts

15 Cites (Scopus)

Resum

A new mechanistic rationalization for the cyclization with hydrogen halides of tautomeric 1,5-dinitriles of general structures (10) (Z = N), (14) (Z = C-CN), (16) (Z = N), and (18) (Z = C-CN) is proposed (Scheme 5). In such rationalization, three factors play a major role on the direction of cyclization: Position of the equilibrium of the tautomeric 1,5-dinitrile system, relative basicity of the cyano groups involved, and planarity of the reaction zone.

Idioma originalAnglès
Pàgines (de-a)739-756
Nombre de pàgines18
RevistaHeterocycles
Volum50
Número2
DOIs
Estat de la publicacióPublicada - 1 d’abr. 1999

Fingerprint

Navegar pels temes de recerca de 'Cyclization of tautomeric 1,5-dinitrile systems with hydrogen halides: A definitive mechanistic rationalization?'. Junts formen un fingerprint únic.

Com citar-ho